What is the standard instruction (SIG) for diltiazem (Cardizem) 2% ointment for the treatment of chronic anal fissures?

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From the Guidelines

The recommended SIG for diltiazem 2% ointment for chronic anal fissures is to apply a pea-sized amount to the affected anal area three times daily for at least 6 weeks, as this duration has been suggested to achieve significant healing rates 1. The primary goal of this treatment is to achieve internal anal sphincter (IAS) relaxation, reducing pain and facilitating the healing process, which is in line with the guidelines for anorectal emergencies 1.

  • Key points to consider when using diltiazem 2% ointment for chronic anal fissures include:
    • Applying the ointment using a gloved finger or applicator, gently inserting it just inside the anal canal and around the anal opening
    • Washing hands thoroughly before and after application
    • Potential mild side effects such as headache or temporary burning upon application
    • Improvement typically seen within 2-3 weeks, but the full course should be completed even if symptoms resolve earlier
    • Follow-up with a healthcare provider if no improvement occurs after 6-8 weeks or if symptoms worsen This treatment approach is supported by recent studies, including a systematic review and meta-analysis that found calcium channel blockers (CCBs) like diltiazem to be more effective than glyceryl trinitrate with less risk of headache and hypotension 1.
  • The use of diltiazem 2% ointment has been associated with healing rates ranging from 65 to 95% and is considered a cost-effective treatment option compared to other non-operative treatments 1.

From the Research

SIG for Diltiazem 2% Ointment

  • The standard instruction for the use of diltiazem 2% ointment for chronic anal fissures is to apply 2 cm (approximately 0.7 g) of the ointment to the anal verge twice daily for eight weeks 2.
  • Alternatively, 8 mg of 2% diltiazem hydrochloride gel (equivalent to 2 cm of gel) can be applied three times daily 3.
  • The application frequency and duration may vary depending on the specific treatment protocol and patient response, with some studies using a 6-week course of twice-daily topical application 4 or a 6-week course of topical diltiazem ointment 5.

Key Considerations

  • Patients should be instructed to report any side effects or symptoms throughout the treatment period 2, 3.
  • The treatment should be monitored for efficacy and safety, with follow-up assessments to evaluate the healing of the fissure and any adverse effects 2, 3, 4, 5.
  • Patients who do not respond to diltiazem treatment may require further treatment, including surgical options such as sphincterotomy 2, 3, 4, 5.

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Research

The role of topical diltiazem in the treatment of chronic anal fissures that have failed glyceryl trinitrate therapy.

Colorectal disease : the official journal of the Association of Coloproctology of Great Britain and Ireland, 2002

Research

Successful treatment of chronic anal fissure with diltiazem gel.

Colorectal disease : the official journal of the Association of Coloproctology of Great Britain and Ireland, 2002

Research

The long-term results of diltiazem treatment for anal fissure.

International journal of clinical practice, 2006

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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