What are the neurologic side effects of Zepbound (Lokelma)?

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Last updated: May 8, 2025View editorial policy

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From the Research

Zepbound (tirzepatide) can cause several neurologic side effects, including headache, dizziness, and fatigue, with the most recent and highest quality study 1 not specifically reporting on neurologic side effects, but previous studies 2, 3, 4, 5 indicating that these effects are generally mild to moderate and may diminish over time.

Common Neurologic Side Effects

  • Headache
  • Dizziness
  • Fatigue
  • Paresthesia (tingling sensations)
  • Changes in taste perception

Serious but Rare Neurologic Effects

  • Hypoglycemia, which can lead to confusion, weakness, or even loss of consciousness if severe
  • Attention difficulties and memory issues in some patients

Management of Neurologic Side Effects

If you experience persistent or severe neurologic symptoms while taking Zepbound, contact your healthcare provider immediately. The neurologic effects are believed to be related to the medication's impact on GLP-1 and GIP receptors in the brain, as these hormones have effects beyond just regulating blood glucose and can influence neural function. Starting with the lowest dose and gradually increasing as tolerated may help minimize these side effects. It is essential to weigh the benefits of Zepbound in improving glycemic control and weight loss against the potential risks of neurologic side effects, prioritizing morbidity, mortality, and quality of life as the primary outcomes 1.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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