What are the medications to naturally reduce hypercholesterolemia (high cholesterol)?

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Last updated: May 12, 2025View editorial policy

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From the Guidelines

Plant sterols and stanols (2 grams daily) are the most effective natural supplements to reduce cholesterol levels, as they can decrease total and LDL cholesterol levels by 9% to 20%. Several natural supplements can help reduce cholesterol levels, including:

  • Red yeast rice (typically 1200-2400 mg daily) which contains natural statins that lower LDL cholesterol 1
  • Plant sterols and stanols (2 grams daily) which block cholesterol absorption in the intestines 1
  • Soluble fiber supplements like psyllium (10-25 grams daily) which bind to cholesterol in the digestive system 1
  • Fish oil supplements (1-4 grams daily of EPA and DHA) which can reduce triglycerides and slightly increase HDL 1
  • Niacin (vitamin B3, 1-3 grams daily) which can lower LDL and raise HDL but should be started at low doses to minimize flushing 1
  • Berberine (500 mg 2-3 times daily) which works similarly to prescription medications by increasing LDL receptors

These supplements work best alongside lifestyle changes like a heart-healthy diet rich in fruits, vegetables, whole grains, and lean proteins, regular exercise, weight management, and avoiding smoking. Always consult with a healthcare provider before starting any supplement regimen, especially if you're taking other medications, as some natural products can interact with prescription drugs.

From the Research

Drugs to Naturally Reduce Cholesterol

  • Plant sterols and stanols have been shown to effectively lower LDL cholesterol levels in hypercholesterolemic, diabetic, and healthy human volunteers 2, 3, 4
  • The hypocholesterolemic effects of plant sterols and stanols are possibly due to their interference with the uptake of both dietary and biliary cholesterol from the intestinal tract 2, 5
  • Studies have demonstrated that unesterified plant sterols and stanols lower LDL-cholesterol concentrations equivalently in hypercholesterolemic persons by suppressing cholesterol absorption 3
  • The LDL-cholesterol-lowering effect of plant sterols and stanols continues to increase up to intakes of approximately 3 g/d to an average effect of 12% 4
  • In addition to lowering LDL cholesterol, plant sterols and stanols may also have beneficial effects on other lipid variables, such as apolipoprotein (apo) B/apoAI ratio, and in some studies, high-density lipoprotein cholesterol (HDL-C) and triglycerides (TG) 6
  • Sitosterol, a type of plant sterol, has been shown to be effective in lowering plasma LDL-C concentrations and may be a useful dietary supplement for the lowering of plasma cholesterol 5

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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