Is hydralazine safe to administer in patients with acute liver failure?

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Last updated: May 18, 2025View editorial policy

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From the Research

Hydralazine should be avoided in patients with acute liver failure due to the risk of worsening liver dysfunction and potential for severe adverse effects, as evidenced by a recent case report of hydralazine-induced fulminant liver failure requiring liver transplant 1.

Key Considerations

  • Hydralazine is metabolized by the liver and can accumulate in patients with impaired liver function, leading to increased risk of adverse effects such as hypotension, tachycardia, headache, and fluid retention.
  • The drug has been associated with rare cases of drug-induced liver injury, which could potentially worsen existing liver dysfunction 2, 3.
  • Alternative antihypertensives that are less dependent on hepatic metabolism, such as certain calcium channel blockers or nitrates, might be safer options in acute liver failure.

Management of Acute Liver Failure

  • Optimal management begins with identifying that liver failure is indeed present and its etiology, since outcomes and the need for transplantation vary widely across the different etiologies 4.
  • Management involves optimizing fluid balance and cardiovascular support, including the use of continuous renal replacement therapy, vasopressors, and pulmonary ventilation.
  • Early evaluation for liver transplantation is advised particularly for acetaminophen toxicity, which evolves so rapidly that delay is likely to lead to death.

Monitoring and Precautions

  • Close monitoring of blood pressure, heart rate, and liver function tests is crucial if hydralazine must be used in patients with acute liver failure.
  • Patients should be closely monitored for signs of worsening liver dysfunction, such as increased liver enzymes, coagulopathy, and encephalopathy.
  • Alternative treatments, such as liver support devices and/or agents that improve hepatocyte regeneration, may be considered in the future 4.

References

Research

Hydralazine-Induced Fulminant Liver Failure Requiring Urgent Liver Transplant: Common Drug With Rare Complication.

Experimental and clinical transplantation : official journal of the Middle East Society for Organ Transplantation, 2023

Research

Hydralazine-induced cholestatic hepatitis.

American journal of therapeutics, 2009

Research

Management of Acute Liver Failure: Update 2022.

Seminars in liver disease, 2022

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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