Does Niacin (Nicotinic Acid) cause tongue swelling?

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Last updated: February 7, 2025View editorial policy

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From the Guidelines

Niacin (Nicotinic Acid) does not have a well-established association with tongue swelling.

Adverse Effects of Niacin

  • The provided evidence primarily discusses the use of niacin in the context of lowering LDL cholesterol and raising HDL cholesterol, as well as its side effects such as skin flushing, hepatotoxicity, hyperuricemia, and hyperglycemia 1.
  • None of the evidence directly links niacin to tongue swelling, suggesting that this is not a commonly recognized or reported side effect.

Safety Recommendations for Niacin

  • The 2013 ACC/AHA guideline on the treatment of blood cholesterol recommends monitoring patients on niacin for adverse effects such as hepatotoxicity, hyperglycemia, and hyperuricemia, but does not mention tongue swelling as a potential side effect 1.
  • The guideline also suggests starting niacin at a low dose and titrating up to a higher dose to minimize adverse effects, but again, does not mention tongue swelling 1.

Conclusion Based on Available Evidence

Given the lack of evidence linking niacin to tongue swelling, it is reasonable to conclude that niacin is not typically associated with this side effect. However, as with any medication, patients should be monitored for any unusual or unexpected side effects, including tongue swelling, and healthcare providers should exercise caution when prescribing niacin, especially in patients with a history of adverse reactions to medications 1.

From the FDA Drug Label

The following additional adverse reactions have been identified during post-approval use of niacin extended-release: Hypersensitivity reactions, including anaphylaxis, angioedema, urticaria, flushing, dyspnea, tongue edema, larynx edema, face edema, peripheral edema, laryngismus, and vesiculobullous rash;

Tongue swelling (also known as tongue edema) is a reported adverse reaction in the postmarketing experience of niacin extended-release, as stated in the drug label 2.

From the Research

Niacin and Tongue Swelling

  • There is no direct evidence in the provided studies that suggests niacin (nicotinic acid) causes tongue swelling 3, 4, 5, 6, 7.
  • The studies primarily focus on the effects of niacin on lipid metabolism, cardiovascular health, and skin conditions, but do not mention tongue swelling as a potential side effect.
  • Common side effects of niacin mentioned in the studies include cutaneous flushing, gastrointestinal disturbances, and hepatotoxicity 3, 5, but tongue swelling is not listed as a known side effect.
  • It is possible that tongue swelling may be a rare or undocumented side effect of niacin, but based on the available evidence, there is no clear link between niacin and tongue swelling.

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Research

A Second Look at Niacin.

Skinmed, 2023

Research

[Niacin in therapy].

Postepy higieny i medycyny doswiadczalnej (Online), 2007

Research

Niacin, an old drug with a new twist.

Journal of lipid research, 2013

Research

Niacin dosing: relationship to benefits and adverse effects.

Current atherosclerosis reports, 2000

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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