What are the common side effects of terbutaline?

Medical Advisory BoardAll articles are reviewed for accuracy by our Medical Advisory Board
Educational purpose only • Exercise caution as content is pending human review
Article Review Status
Submitted
Under Review
Approved

Last updated: September 6, 2025View editorial policy

Personalize

Help us tailor your experience

Which best describes you? Your choice helps us use language that's most understandable for you.

Common Side Effects of Terbutaline

Terbutaline commonly causes tremor, tachycardia, anxiety, palpitations, and nervousness as side effects due to its beta-adrenergic stimulating properties. 1

Primary Side Effect Profile

Terbutaline is a selective beta-2 agonist used primarily as a bronchodilator for asthma treatment. Its side effects are primarily related to its sympathomimetic activity:

Cardiovascular Effects

  • Heart rate increases: Tachycardia is common and dose-dependent 1, 2
  • Palpitations and chest pain 1
  • Blood pressure changes: Typically increases systolic while decreasing diastolic pressure 2
  • Cardiac arrhythmias in susceptible patients 1
  • Myocardial ischemia (rare but serious) 1

Neurological/Musculoskeletal Effects

  • Tremor: Most common side effect, dose-dependent 3
  • Anxiety and nervousness 1
  • Headache 4
  • Dizziness 5
  • Seizures (rare): Case reports exist of focal seizures in pediatric patients 5

Metabolic Effects

  • Transient hyperglycemia: Blood glucose increases 2
  • Hypokalemia: Due to intracellular potassium shifting 1, 6
  • Potential worsening of diabetes in susceptible patients 1

Special Considerations

Pregnancy Concerns

While not directly related to the question about common side effects, it's important to note that terbutaline has serious risks when used for tocolysis (delaying preterm labor):

  • Pulmonary edema (0.32% incidence) 7
  • Cardiac arrhythmias 1
  • Myocardial ischemia 1
  • The FDA has explicitly warned against using terbutaline for tocolysis due to serious maternal and fetal risks 8

Pediatric Considerations

  • In appropriate doses (2.5 mg orally for children 7-14 years weighing 25-50 kg), terbutaline has shown minimal cardiovascular side effects 9
  • However, terbutaline is not recommended for patients under 12 years due to insufficient safety data 1

Drug Interactions

  • Beta-blockers: Can block bronchodilator effects and potentially cause severe bronchospasm 1
  • MAOIs and tricyclic antidepressants: May potentiate cardiovascular effects 6
  • Non-potassium sparing diuretics: May worsen ECG changes and hypokalemia 6

Comparative Safety Profile

When administered by inhalation rather than systemically, terbutaline produces similar bronchodilation with significantly fewer systemic side effects 3, making the inhaled route preferable when possible.

The side effect profile is similar to other beta-2 agonists, though some studies report that terbutaline may cause more frequent tremor than other agents in this class 4.

References

Research

Cardiovascular and metabolic effects of terbutaline.

Journal of clinical and hospital pharmacy, 1982

Research

Comparison of infused and inhaled terbutaline in patients with asthma.

Scandinavian journal of respiratory diseases, 1976

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Tocolysis Guidelines

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

Have a follow-up question?

Our Medical A.I. is used by practicing medical doctors at top research institutions around the world. Ask any follow up question and get world-class guideline-backed answers instantly.