What is the recommended dose of octreotide (somatostatin analogue) per kilogram?

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Octreotide Per Kilogram Dosing

For pediatric sulfonylurea poisoning, octreotide should be dosed at 1-1.5 μg/kg IV or SC, followed by 2-3 additional doses every 6 hours. 1

Weight-Based Dosing Context

The per-kilogram dosing of octreotide is primarily established and recommended in pediatric populations, particularly for sulfonylurea-induced hypoglycemia. 1 This represents the most clearly defined weight-based dosing protocol in the medical literature.

Pediatric Sulfonylurea Poisoning Protocol

  • Initial dose: 1-1.5 μg/kg IV or SC 1
  • Maintenance: Repeat doses every 6 hours for 2-3 additional doses 1
  • Concurrent therapy: IV dextrose should be gradually tapered during octreotide treatment 1
  • Clinical context: This dosing was effective in 14 pediatric patients who ingested sulfonylureas, with 50% experiencing recurrent hypoglycemia requiring additional doses 1

Important Caveat for Pediatric Use

  • One pediatric patient developed hypertension and apnea 30 minutes after IV octreotide, though the causal relationship remains unclear 1
  • Recurrent hypoglycemia occurred in 50% of pediatric cases despite octreotide therapy, necessitating additional doses and IV dextrose 1

Adult Dosing (Not Weight-Based)

In contrast to pediatric protocols, adult dosing is typically fixed rather than weight-based:

Standard Adult Dosing Regimens

  • Short-acting subcutaneous: 50-100 μg SC every 8 hours, with doses ranging up to 150-250 μg three times daily for breakthrough symptoms 2, 3
  • IV drip: 50 μg/hour continuous infusion, typically preceded by 50 μg IV bolus 4
  • Long-acting release (LAR): 20-30 mg intramuscularly every 4 weeks 2

Carcinoid Crisis Prevention

  • Perioperative dosing: 50 μg/hour IV infusion starting 12 hours before procedures and continuing 24-48 hours after 4, 3, 5

Dose Escalation in Adults

  • Clinical benefit may occur with doses as low as 50 μg, but some patients require up to 1500 μg/day 3
  • For refractory chemotherapy-induced diarrhea, doses can be titrated up to 500 μg three times daily 4, 3
  • In acromegaly studies, doses up to 3000 μg/day have been administered without serious adverse effects, though doses above 800 μg/day rarely provide additional benefit 6, 7

Clinical Pitfall

The critical distinction: Weight-based dosing (μg/kg) is established for pediatric sulfonylurea poisoning, while adult dosing across all other indications uses fixed doses regardless of body weight. 1, 2 Do not extrapolate pediatric weight-based dosing to adult populations for neuroendocrine tumors, carcinoid syndrome, or other standard indications.

References

Research

Octreotide for the treatment of sulfonylurea poisoning.

Clinical toxicology (Philadelphia, Pa.), 2012

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Octreotide Dosage and Administration

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Initial Octreotide Drip Dosage

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Octreotide Therapy for Neuroendocrine Tumors

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Research

Octreotide, a new somatostatin analogue.

Clinical pharmacy, 1989

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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