What is the dosage and usage of Cisatracurium (a neuromuscular blocking agent) for tracheal intubation and surgery?

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Cisatracurium Dosing and Usage for Tracheal Intubation and Surgery

Initial Intubating Doses

For tracheal intubation, administer cisatracurium 0.15-0.2 mg/kg IV, with the 0.2 mg/kg dose providing superior intubation conditions at 1.5 minutes compared to 2 minutes with 0.15 mg/kg. 1

Standard Dosing Protocol

  • 0.15 mg/kg (3 x ED95): Produces good to excellent intubation conditions in 2 minutes with a clinically effective duration of 55 minutes (range: 44-74 minutes) 1

  • 0.2 mg/kg (4 x ED95): Produces excellent intubation conditions in 1.5 minutes with a clinically effective duration of 61 minutes (range: 41-81 minutes), and is the preferred dose for optimal intubation conditions 1, 2

  • Both doses achieve good or excellent intubation conditions in over 90% of patients when used with propofol/nitrous oxide/oxygen or thiopental-based induction techniques 1, 2

Mechanism and Rationale

  • Cisatracurium is a benzylisoquinolinium non-depolarizing neuromuscular blocking agent that competitively binds cholinergic receptors at the motor end plate 3

  • The use of muscle relaxants like cisatracurium reduces poor intubating conditions from 24.6% to 4.1% and decreases pharyngeal/laryngeal injury from 18.7-22.6% to 9.7% 4, 3

Maintenance Dosing During Surgery

Administer 0.03 mg/kg cisatracurium for maintenance of neuromuscular blockade, which sustains block for approximately 20 minutes. 1

Maintenance Timing

  • First maintenance dose typically required 40-50 minutes after initial 0.15 mg/kg dose 1

  • First maintenance dose typically required 50-60 minutes after initial 0.2 mg/kg dose 1

  • Subsequent maintenance doses should be guided by clinical criteria and train-of-four (TOF) monitoring 1

Continuous Infusion Alternative

  • After initial bolus, cisatracurium can be administered by continuous infusion for extended procedures in adults and children ≥2 years 1

  • Infusion rates should be individualized based on TOF monitoring 1

Special Population Adjustments

Elderly and Renal Dysfunction Patients

  • Extend the interval between cisatracurium administration and intubation attempt due to slower onset times in these populations 1

  • No dose adjustment necessary due to organ-independent Hofmann elimination 3, 1

Obese Patients

  • Calculate cisatracurium dose based on ideal body weight, not actual body weight 3

Pediatric Dosing

  • Children 2-12 years: 0.1-0.15 mg/kg produces maximum block in 2.8-3 minutes with 28-36 minutes of clinically effective block 1

  • Infants 1-23 months: 0.15 mg/kg produces maximum block in approximately 2 minutes with 43 minutes of clinically effective block 1

Volatile Anesthetic Interactions

Isoflurane or enflurane at 1.25 MAC prolongs the duration of cisatracurium, requiring less frequent or lower maintenance doses. 1

  • Initial 15-30 minutes of volatile agent exposure has minimal effect on initial dose requirements 1

  • No initial dose adjustment needed when cisatracurium is administered shortly after volatile agent initiation 1

  • In prolonged procedures with volatile anesthetics, reduce maintenance dose frequency or amount 1

  • No dose adjustment required with propofol anesthesia 1

Monitoring Requirements

Use peripheral nerve stimulator monitoring to optimize cisatracurium dosing and minimize risk of overdosage or underdosage. 1

  • Train-of-four monitoring is mandatory throughout anesthesia 5

  • Target TOF ratio ≥0.9 at adductor pollicis to eliminate residual neuromuscular blockade 5

  • Recovery to TOF ratio >0.7 occurs within 34-85 minutes after discontinuation 3

Reversal Considerations

Administer neostigmine 0.05 mg/kg plus glycopyrrolate 10 mcg/kg when tactile TOF count reaches 2 or more to ensure TOF ratio >0.7 in the PACU. 6

  • When neostigmine reversal is delayed until TOF count ≥2, postoperative weakness (TOF <0.7) should be rare 6

  • At 10 minutes post-reversal, expect TOF ratios of approximately 0.72-0.76 6

  • By 15 minutes post-reversal, nearly all patients achieve TOF ratio ≥0.7 6

Critical Pitfalls and Caveats

ICU Patients Require Higher Doses

  • ICU patients require significantly higher cumulative doses (10 ± 4.7 ED95) compared to elective surgery patients (3 ± 0.3 ED95) due to altered pharmacodynamics 7

  • The standard 0.15 mg/kg dose fails to achieve complete paralysis in ICU patients, requiring repeated boluses 7

  • Neuromuscular monitoring is essential in ICU settings due to unpredictable response 7

Laryngeal Muscle Considerations

  • Cisatracurium has slower onset at laryngeal muscles (196 seconds with 0.1 mg/kg) compared to equipotent atracurium doses due to higher potency 8

  • The 0.15 mg/kg dose achieves 92% maximum blockade at the larynx, while 0.2 mg/kg achieves 100% blockade in 148 seconds 8

Administration Route

  • Cisatracurium must only be administered intravenously 1

  • Contains benzyl alcohol—use caution in neonates and infants 1

References

Research

Evaluation of cisatracurium, a new neuromuscular blocking agent, for tracheal intubation.

Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1996

Guideline

Cisatracurium Use in Clinical Settings

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Muscle Relaxants in Anesthesia

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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