Is Tislelizumab (generic name) approved for head and neck cancers?

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Last updated: December 17, 2025View editorial policy

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Tislelizumab Approval Status for Head and Neck Cancers

Yes, tislelizumab is approved and strongly recommended for head and neck cancers, specifically for recurrent or metastatic nasopharyngeal carcinoma as first-line treatment in combination with gemcitabine and cisplatin. 1

Approved Indication

Tislelizumab, combined with gemcitabine and cisplatin, should be offered as first-line treatment for patients with recurrent or metastatic nasopharyngeal cancer (evidence quality: high; strength of recommendation: strong). 1, 2

Key Clinical Details:

  • Dosing regimen: 200 mg intravenously every 3 weeks for 4-6 cycles in combination with chemotherapy, followed by tislelizumab maintenance until disease progression (up to 2 years). 2, 3
  • Chemotherapy backbone: Gemcitabine 1,000 mg/m² on days 1 and 8, plus cisplatin 80 mg/m² on day 1, every 21 days. 2
  • PD-L1 testing not required: Clinical benefit is observed regardless of PD-L1 expression status. 2

Evidence Supporting Use

The recommendation is based on high-quality evidence demonstrating:

  • Progression-free survival: 11.7 months with tislelizumab plus chemotherapy versus 8.0 months with chemotherapy alone (HR 0.52,95% CI 0.36-0.74). 2
  • Overall survival benefit: 40% reduction in risk of death (HR 0.603,95% CI 0.364-0.997), with median OS not reached in the tislelizumab arm versus 33.7 months with placebo. 2
  • Efficacy independent of PD-L1 status: Benefit demonstrated in both PD-L1-negative and PD-L1-positive subgroups. 2

Alternative Options

If tislelizumab is unavailable, pembrolizumab or nivolumab may be offered with gemcitabine and cisplatin, though this carries a lower evidence quality and weaker recommendation. 1, 2

Other Head and Neck Cancer Subtypes

For non-nasopharyngeal head and neck squamous cell carcinoma (HNSCC), tislelizumab is not specifically mentioned in current ASCO guidelines. The preferred agents for recurrent or metastatic HNSCC are:

  • Pembrolizumab (monotherapy or with platinum/fluorouracil) for CPS ≥ 1. 1
  • Nivolumab for platinum-refractory disease. 1

Real-world data from 39 patients with HNSCC or nasopharyngeal carcinoma treated with tislelizumab showed promising efficacy (ORR 86.7% in neoadjuvant setting, 60% in salvage therapy) with acceptable tolerability. 4 However, this does not constitute regulatory approval for non-nasopharyngeal HNSCC.

Safety Profile

Tislelizumab demonstrates an acceptable safety profile with most adverse events ≤ grade 2, though grade 4 enteritis has been reported. 4 Common adverse effects include fatigue, anemia, and decreased neutrophil count. 5

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Toripalimab Treatment for Nasopharyngeal Carcinoma

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Tislelizumab Dosing for Cancer Treatment

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Research

Tislelizumab: A Modified Anti-tumor Programmed Death Receptor 1 Antibody.

Cancer control : journal of the Moffitt Cancer Center, 2022

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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