Can acephate cause hemolysis?

Medical Advisory BoardAll articles are reviewed for accuracy by our Medical Advisory Board
Educational purpose only • Exercise caution as content is pending human review
Article Review Status
Submitted
Under Review
Approved

Last updated: December 18, 2025View editorial policy

Personalize

Help us tailor your experience

Which best describes you? Your choice helps us use language that's most understandable for you.

Can Acephate Cause Hemolysis?

No, acephate does not cause hemolysis based on available evidence. The provided research on acephate toxicity does not document hemolytic anemia as a recognized adverse effect of this organophosphate insecticide.

Evidence from Acephate Exposure Studies

The available human and animal data on acephate exposure focuses on its organophosphate toxicity profile without any mention of hemolysis:

  • Human case reports of acute acephate ingestion document cholinergic toxicity (muscarinic and nicotinic signs), severely depressed cholinesterase activity, and prolonged intensive care requirements, but no hemolysis was reported 1

  • Occupational exposure studies in workers with significant acephate exposure (urinary levels 1-10 mg/L) showed cholinesterase depression in some cases but no hemolytic effects 2

  • Animal toxicity studies demonstrated thiamine depletion, altered carbohydrate metabolism, and glycogen depletion, but did not report hemolysis 3

Mechanism of Acephate Toxicity

Acephate's toxicity operates through organophosphate mechanisms, not oxidative stress pathways that would cause hemolysis:

  • Acephate is metabolized to methamidophos, a potent anticholinesterase agent, though this conversion is limited in humans 1, 2

  • The primary toxic effects involve cholinesterase inhibition, not red blood cell membrane damage 1

  • Unlike medications that cause hemolysis in G6PD deficiency (such as dapsone, primaquine, or methylene blue), acephate is not listed among oxidant drugs that trigger hemolytic crises 4, 5

Clinical Distinction

It is critical to distinguish acephate from medications that do cause hemolysis:

  • Drug-induced hemolytic anemia is well-documented with certain cephalosporins (like cefotetan), which can cause severe acute hemolysis with hemoglobinuria and renal failure 6

  • Oxidant medications contraindicated in G6PD deficiency (dapsone, methylene blue, primaquine) cause hemolysis through oxidative stress mechanisms 4

  • Acephate does not share these oxidative properties or hemolytic risk profiles

Clinical Management of Acephate Toxicity

When managing acephate poisoning, focus on cholinergic toxicity rather than hemolysis:

  • Monitor for cholinergic signs (salivation, lacrimation, urination, defecation, bronchospasm, bradycardia) 1

  • Check red blood cell and plasma cholinesterase levels 2

  • Treat with atropine and pralidoxime as needed for organophosphate poisoning 1

  • Do not implement hemolysis monitoring protocols unless another concurrent cause is suspected

References

Research

Urinary elimination kinetics of acephate and its metabolite, methamidophos, in urine after acute ingestion.

Journal of medical toxicology : official journal of the American College of Medical Toxicology, 2009

Research

Biological monitoring of human exposure to acephate.

Archives of environmental contamination and toxicology, 1990

Guideline

Medications Contraindicated in G6PD Deficiency

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Precautions in G6PD Deficiency

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

Have a follow-up question?

Our Medical A.I. is used by practicing medical doctors at top research institutions around the world. Ask any follow up question and get world-class guideline-backed answers instantly.