Is losartan (angiotensin II receptor antagonist) efficacious when administered twice daily?

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Last updated: April 8, 2025View editorial policy

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From the FDA Drug Label

The studies allowed comparisons of two doses (50 to 100 mg/day) as once-daily or twice-daily regimens, comparisons of peak and trough effects, and comparisons of response by gender, age, and race. Twice-daily dosing at 50 mg to 100 mg/day gave consistently larger trough responses than once-daily dosing at the same total dose.

  • Efficacy: Losartan is efficacious when given twice daily, as twice-daily dosing at 50 mg to 100 mg/day gave consistently larger trough responses than once-daily dosing at the same total dose.
  • Dosage: The appropriate dosage for twice-daily administration is 50 mg to 100 mg/day, divided into two doses. 1

From the Research

Losartan should not be given twice daily, as once-daily dosing is the standard and appropriate regimen, providing 24-hour blood pressure control with a single dose. The usual adult dosage ranges from 25-100 mg once daily, with 50 mg being a common starting dose for hypertension. According to the most recent and highest quality study, 2, there were no differences in systolic/diastolic blood pressure between twice-daily and once-daily dosing, with absolute differences in mean systolic blood pressure ranging from -1.8 to 0.7 mmHg and diastolic blood pressure ranging from -1.1 to 0.1 mmHg. This study suggests that once-daily dosing is sufficient and effective for blood pressure control.

Some key points to consider when prescribing losartan include:

  • The active metabolite of losartan has a half-life of 6-9 hours, providing 24-hour blood pressure control with once-daily administration.
  • While some patients might benefit from divided dosing in specific circumstances, this is not routinely recommended or necessary.
  • The once-daily dosing schedule improves medication adherence and maintains consistent blood pressure control throughout the day.
  • If blood pressure control is inadequate with maximum once-daily dosing (100 mg), adding a different antihypertensive medication rather than splitting the losartan dose is generally preferred.
  • Patients should take losartan at the same time each day to maintain consistent blood levels and therapeutic effect.

It's also worth noting that the study 2 found no improved effectiveness or safety of twice-daily dosing compared to once-daily dosing, which further supports the use of once-daily dosing as the standard regimen.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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