What is the landmark trial that showed no benefit of azathioprine with Tumor Necrosis Factor (TNF)-alpha agonists, such as adalimumab (adalimumab), in the treatment of inflammatory bowel disease?

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Landmark Trial: UC-SUCCESS

The UC-SUCCESS trial is the landmark study that demonstrated combination therapy of infliximab plus azathioprine was superior to either monotherapy in ulcerative colitis, achieving 39.7% corticosteroid-free remission at week 16 compared to 22.1% with infliximab alone and 23.7% with azathioprine alone. 1

Key Trial Details

The UC-SUCCESS trial was a randomized, double-blind study in anti-TNF-naïve adults with moderate to severe ulcerative colitis that compared three arms: 1

  • Infliximab monotherapy (5 mg/kg at weeks 0,2,6, and 14)
  • Azathioprine monotherapy (2.5 mg/kg daily)
  • Combination therapy (infliximab plus azathioprine)

The trial enrolled 239 patients and was terminated prematurely before reaching enrollment targets, which limited the ability to complete the planned maintenance phase. 2, 1

Primary Outcome Results

Corticosteroid-free remission at week 16 (the primary endpoint): 1

  • Combination therapy: 39.7% (31/78 patients)
  • Infliximab monotherapy: 22.1% (17/77 patients) - p=0.017 vs combination
  • Azathioprine monotherapy: 23.7% (18/76 patients) - p=0.032 vs combination

Secondary Outcomes

Mucosal healing at week 16 showed: 1

  • Combination therapy: 62.8% (49/78 patients)
  • Infliximab monotherapy: 54.6% (42/77 patients) - p=0.295 vs combination
  • Azathioprine monotherapy: 36.8% (28/76 patients) - p=0.001 vs combination

The combination therapy demonstrated statistically significant superiority over azathioprine monotherapy for mucosal healing, though the difference versus infliximab monotherapy did not reach statistical significance. 1

Important Clarification About Your Question

Your question contains a critical error: The UC-SUCCESS trial showed benefit of adding azathioprine to infliximab, not "no benefit." 1 There is no landmark trial showing no benefit of combination therapy with TNF-alpha antagonists and azathioprine in ulcerative colitis.

Current Guideline Recommendations Based on UC-SUCCESS

The 2020 AGA guidelines conditionally suggest combining TNF-α antagonists with thiopurines or methotrexate rather than biologic monotherapy in moderate-severe ulcerative colitis, based primarily on the UC-SUCCESS trial results. 2

However, the guidelines acknowledge this is a conditional recommendation with low-quality evidence because: 2

  • The trial was terminated prematurely
  • No maintenance phase data were completed
  • Evidence for non-infliximab TNF antagonists is extrapolated (indirect evidence)
  • Newer biologics may have lower immunogenicity than infliximab

Safety Considerations

Serious infections occurred in only 2 patients in UC-SUCCESS (one receiving infliximab monotherapy, one receiving azathioprine monotherapy), though combination therapy with anti-TNF agents and thiopurines generally increases risk of opportunistic infections and malignancy. 2, 1

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Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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