What is the use of benzocaine (Tessalon) pearls?

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From the Guidelines

Benzocaine, also known as Tessalon pearls, is used as a pharyngeal anesthetic agent to facilitate upper endoscopic procedures and reduce discomfort during medical procedures.

Key Points

  • Benzocaine has an onset of 5 minutes and a duration of 15-45 minutes 1
  • It is used as an adjunct to moderate sedation to reduce discomfort and facilitate procedures such as upper endoscopy 1
  • However, benzocaine has been associated with a potentially life-threatening adverse event known as methemoglobinemia, which requires prompt diagnosis and treatment with intravenous methylene blue 1

Usage and Precautions

  • Benzocaine can be used for topical anesthesia in office-based dermatologic surgery, but caution must be taken to avoid adverse events such as methemoglobinemia 1
  • It is essential to be aware of the potential risks and take necessary precautions when using benzocaine, especially in patients with certain medical conditions or taking specific medications 1

From the Research

Use of Benzocaine (Tessalon) Pearls

  • Benzocaine pearls, also known as Tessalon Perles, are used for rapid oral anesthesia in preparation for awake intubations 2.
  • They can provide effective topical oral anesthesia, with a shorter time to obtain loss of the gag response compared to other methods 2.
  • Benzocaine lozenges, which contain benzocaine, are also used in the treatment of uncomplicated sore throat, providing superior pain relief compared to placebo lozenges 3.
  • The use of benzocaine spray for throat pain has been reported to lead to suspected methemoglobinemia, a rare complication associated with benzocaine 4.
  • Tessalon Perles have also been involved in cases of overdose, resulting in cardiac arrest and residual blindness 5, and fatalities 6.

Clinical Applications

  • Awake intubations: Benzocaine pearls can be used to provide rapid and reliable oropharyngeal anesthesia in preparation for awake intubations 2.
  • Sore throat treatment: Benzocaine lozenges can be used to reduce painful pharyngeal discomfort in patients with uncomplicated sore throat 3.
  • Local anesthesia: Benzocaine can be used as a local anesthetic to provide rapid pain relief 4.

Safety Considerations

  • Methemoglobinemia: Benzocaine can cause methemoglobinemia, a rare complication that can lead to respiratory distress and potentially fatal outcomes if not promptly diagnosed and treated 4.
  • Overdose: Tessalon Perles can be involved in cases of overdose, resulting in cardiac arrest and residual blindness 5, and fatalities 6.

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Research

Rapid oral anesthesia for awake intubation.

Journal of clinical anesthesia, 1992

Research

Efficacy of a benzocaine lozenge in the treatment of uncomplicated sore throat.

European archives of oto-rhino-laryngology : official journal of the European Federation of Oto-Rhino-Laryngological Societies (EUFOS) : affiliated with the German Society for Oto-Rhino-Laryngology - Head and Neck Surgery, 2012

Research

Two fatalities resulting from Tessalon (benzonatate).

Veterinary and human toxicology, 1986

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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