What is the comparison of adherence between long-acting injectable (LAI) and oral medications in outpatient settings?

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From the Guidelines

Long-acting injectable antipsychotics are recommended over oral medications for outpatient adherence due to their ability to eliminate daily medication administration and reduce relapse rates by 20-30%. This recommendation is based on the most recent and highest quality evidence available, including guidelines from the British Journal of Psychiatry 1 and case vignettes that illustrate the benefits of long-acting injections in patients with a history of non-adherence 1.

Key Points to Consider

  • Long-acting injectable antipsychotics, such as paliperidone palmitate, risperidone, aripiprazole, and haloperidol decanoate, provide steady plasma levels and reduce side effects, leading to improved adherence.
  • Patients should be stabilized on the oral version of the medication before transitioning to the injectable form, and most LAIs require initial loading doses followed by regular maintenance injections.
  • Regular contact with healthcare providers for injections creates opportunities for intervention if problems arise, and LAIs may be particularly beneficial for patients with a history of recurrent relapses related to partial or full non-adherence.
  • However, LAIs may not be suitable for all patients due to cost considerations, needle phobia, or personal preferences for autonomy in medication management.

Implementation and Monitoring

  • Healthcare providers should consider long-acting injection antipsychotic medication for patients who have a history of non-adherence or recurrent relapses, as it can be a valuable treatment option to improve adherence and reduce relapse rates.
  • Patients should be closely monitored during the transition to LAIs, and regular follow-up appointments should be scheduled to assess treatment efficacy and address any concerns or side effects.
  • As noted in the guidelines, depot preparations should be offered as a treatment option where a service user expresses a preference for such treatment because of its convenience or as part of a treatment plan in which avoidance of covert non-adherence to the antipsychotic regimen is a clinical priority 1.

From the Research

Long Acting Injectable vs Oral Outpatient Adherence

  • Long-acting injectable (LAI) antipsychotic medications can help improve treatment adherence in patients with schizophrenia and bipolar disorder 2.
  • Rates of adherence to treatment in patients with schizophrenia and bipolar disorder are low, and individualizing care can help improve this 2.
  • A personalized intervention to address adherence barriers combined with LAI can improve recovery outcomes in high-risk individuals with bipolar disorder 3.
  • The proportion of missed medications in the past week significantly improved from 50.1% to 16.9% when using LAI antipsychotic medication plus customized adherence enhancement in poorly adherent individuals with bipolar disorder 3.

Comparison of LAI and Oral Formulations

  • There is little evidence on comparisons between LAIs and their oral mother compounds, and even less concerning effectiveness comparisons between different depots 4.
  • LAI antipsychotics have a clear advantage over placebo regarding relapse prevention and symptom reduction, but their effectiveness compared to oral formulations is not well established 4.
  • Paliperidone, a second-generation antipsychotic, has demonstrated efficacy in the reduction of acute schizophrenia symptoms and clinical benefits were maintained also in the long-term treatments, both as an extended-release (ER) oral formulation and a long-acting injectable paliperidone palmitate (PP) formulation 5.

Adherence and Outcomes

  • Improving adherence to antipsychotic medication is crucial for achieving better outcomes in patients with schizophrenia and bipolar disorder 2, 3.
  • Customized adherence enhancement approaches can help improve adherence and outcomes in high-risk individuals with bipolar disorder 3.
  • The use of LAI antipsychotic medication can help reduce the risk of relapse and improve symptom reduction in patients with schizophrenia and bipolar disorder 4, 3.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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