Is hydroxyurea used to treat renal cell carcinoma?

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Last updated: February 18, 2026View editorial policy

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Hydroxyurea is NOT Used to Treat Renal Cell Carcinoma

Hydroxyurea has no role in the modern treatment of renal cell carcinoma and is not recommended by any current clinical practice guidelines. 1, 2

Current Standard Treatment for Metastatic RCC

The established first-line treatments for metastatic renal cell carcinoma are:

  • For intermediate and poor-risk patients: Nivolumab plus ipilimumab (immune checkpoint inhibitors) 2
  • For good and intermediate-risk patients: VEGF-targeted agents including sunitinib, pazopanib, or bevacizumab plus interferon 1, 2
  • For poor-prognosis patients: Temsirolimus (mTOR inhibitor) 1

Why Hydroxyurea Is Not Used

Renal cell carcinoma is highly resistant to systemic chemotherapy, and no chemotherapy agent should be considered standard treatment for metastatic disease. 3 The multiple ESMO Clinical Practice Guidelines for RCC from 2012,2014, and 2019 make no mention of hydroxyurea as a treatment option for any stage of renal cell carcinoma. 1

Historical Context Only

While one small phase II study from 1978 reported responses in 5 of 8 patients using a combination regimen that included hydroxyurea with adriamycin, vinblastine, and medroxyprogesterone acetate, this approach was never validated or adopted into clinical practice. 4 The median survival in that study was only 4 months, and this combination therapy has been completely superseded by modern targeted therapies and immunotherapies. 4

Common Pitfall to Avoid

Do not confuse hydroxyurea's established role in sickle cell disease and certain myeloproliferative disorders with any indication for renal cell carcinoma. 1, 5, 6 Hydroxyurea inhibits ribonucleotide reductase and has legitimate uses in other conditions, but RCC's inherent chemoresistance makes it ineffective for this malignancy. 5, 3

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Management of Renal Cell Carcinoma

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Research

Chemotherapy for renal cell carcinoma.

Seminars in oncology, 2000

Research

Hydroxyurea and hydroxamic acid derivatives as antitumor drugs.

Cancer chemotherapy and pharmacology, 2009

Research

Hydroxyurea: an overview.

Journal of biological regulators and homeostatic agents, 1999

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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