What alternative medication is taken if Loperamide (loperamide) does not work for diarrhea?

Medical Advisory BoardAll articles are reviewed for accuracy by our Medical Advisory Board
Educational purpose only • Exercise caution as content is pending human review
Article Review Status
Submitted
Under Review
Approved

Last updated: April 25, 2025View editorial policy

Personalize

Help us tailor your experience

Which best describes you? Your choice helps us use language that's most understandable for you.

From the Guidelines

If loperamide doesn't work for diarrhea, azithromycin is a recommended alternative, given its strong recommendation and high level of evidence for treating moderate travelers’ diarrhea. When considering alternative medications, several options can be evaluated based on the cause and severity of the diarrhea.

  • For moderate travelers’ diarrhea, fluoroquinolones may be used, although with caution due to the emergence of resistance and potential adverse effects 1.
  • Azithromycin is a preferred choice due to its strong recommendation and high level of evidence, making it a suitable option for treating moderate travelers’ diarrhea 1.
  • Rifaximin may also be considered, but with caution, especially in regions with a high risk of invasive pathogens 1. It's crucial to note that the choice of medication should be guided by the severity of symptoms, potential causes, and the patient's medical history.
  • Staying hydrated with electrolyte solutions is essential while taking these medications.
  • If diarrhea persists or is accompanied by severe symptoms, medical attention should be sought to rule out more serious conditions requiring different treatment.

From the Research

Alternative Medications for Diarrhea

If loperamide does not work for diarrhea, other medications can be considered.

  • Bismuth subsalicylate is an alternative option, as seen in a study comparing loperamide with bismuth subsalicylate for the treatment of acute travelers' diarrhea 2.
  • Trimethoprim-sulfamethoxazole can be used for subjects whose condition is not improved with loperamide therapy, as mentioned in a study on acute nondysenteric travelers' diarrhea 2.
  • Antibiotics such as fluoroquinolones, azithromycin, and rifaximin may be used for moderate to severe travelers' diarrhea, with loperamide considered as monotherapy or adjunctive therapy 3.

Considerations for Treatment

When considering alternative medications, it is essential to note the following:

  • Loperamide is effective for painless diarrhea and is considered to be free of abuse potential 4, 5.
  • Bismuth subsalicylate is less effective than loperamide in reducing the average number of unformed bowel movements 6.
  • Antibiotics should be used judiciously, as they may not be necessary for mild cases of travelers' diarrhea 3.

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Research

Travelers' Diarrhea: A Clinical Review.

Recent patents on inflammation & allergy drug discovery, 2019

Research

Loperamide: a pharmacological review.

Reviews in gastroenterological disorders, 2007

Research

Safety and efficacy of loperamide.

The American journal of medicine, 1990

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

Have a follow-up question?

Our Medical A.I. is used by practicing medical doctors at top research institutions around the world. Ask any follow up question and get world-class guideline-backed answers instantly.