What is the role of Zepbound (exenatide) in the treatment of Polycystic Ovary Syndrome (PCOS)?

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Last updated: April 25, 2025View editorial policy

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From the Research

Zepbound (tirzepatide) should not be considered as a first-line treatment for PCOS, but rather as an off-label option for patients with obesity or type 2 diabetes, with lifestyle modifications and metformin being the primary approaches, as supported by the most recent and highest quality study 1.

Key Considerations

  • The most recent study 1 emphasizes the importance of lifestyle interventions, including dietary changes and physical activity, in managing PCOS, which should be the primary approach.
  • Metformin, as discussed in studies 2, 3, and 4, is a well-established treatment for PCOS, particularly for improving insulin sensitivity and regulating menstrual cycles.
  • Zepbound (tirzepatide) may be considered for PCOS patients with obesity or type 2 diabetes, as it can promote weight loss, improve insulin sensitivity, and potentially reduce androgen levels, as seen in other contexts.

Treatment Approach

  • Lifestyle modifications, including a balanced diet and regular physical activity, should be the first-line approach for managing PCOS, as recommended by the most recent study 1.
  • Metformin should be considered for patients with insulin resistance or type 2 diabetes, as it has been shown to improve insulin sensitivity and regulate menstrual cycles 2, 3, and 4.
  • Zepbound (tirzepatide) may be considered as an off-label treatment option for PCOS patients with obesity or type 2 diabetes, with careful monitoring of side effects and blood glucose levels.

Important Considerations

  • Patients should discuss their individual symptoms and goals with their healthcare provider to determine the most appropriate treatment approach.
  • Blood glucose monitoring may be necessary, especially if the patient has diabetes or prediabetes.
  • Common side effects of Zepbound (tirzepatide) include nausea, diarrhea, vomiting, and constipation, which often improve over time.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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