What is the role of Pembrolizumab (pembrolizumab) in breast cancer (breast ca)?

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Last updated: April 29, 2025View editorial policy

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From the Guidelines

Pembrolizumab is recommended for triple-negative breast cancer (TNBC) as neoadjuvant therapy with chemotherapy, followed by adjuvant pembrolizumab for a total treatment duration of approximately one year, as stated in the most recent guideline from 2024 1.

Key Points

  • Pembrolizumab should be administered every 3 weeks throughout the neoadjuvant phase and for nine 3-week cycles during the adjuvant phase, regardless of pCR status 1.
  • The use of dose-dense schedules of chemotherapy, with granulocyte colony-stimulating factor support, should be considered given their documented benefit over non-dose-dense schedules 1.
  • Patients receiving pembrolizumab should be monitored very closely for the risk of immune-related adverse events throughout treatment and following the ESMO CPG for the management of toxicities from immunotherapy 1.
  • For high-risk early-stage TNBC, neoadjuvant treatment is preferred, and pembrolizumab can be given in combination with chemotherapy, unless there are risk factors for excessive ICI-associated immune toxicity 1.

Treatment Considerations

  • The combination of ICIs and olaparib may be considered on an individual basis, but the combination of olaparib and capecitabine in patients with gBRCAm should not be used 1.
  • Patients with residual disease who did not receive ICIs should be offered adjuvant capecitabine for 6-8 cycles 1.
  • The ESMO-MCBS v1.1 score and ESCAT scores can be used to guide treatment decisions, with a score of A indicating a high level of evidence and a strong recommendation for treatment 1.

Monitoring and Follow-up

  • Patients should be monitored for immune-related adverse events, including pneumonitis, colitis, hepatitis, endocrinopathies, and skin reactions 1.
  • Treatment should be continued until disease progression, unacceptable toxicity, or completion of planned therapy 1.

From the Research

Pembrolizumab in Breast Cancer

  • Pembrolizumab has been studied in combination with chemotherapy for the treatment of advanced triple-negative breast cancer, with results showing longer progression-free survival and overall survival compared to chemotherapy alone in patients with tumors expressing PD-L1 with a combined positive score (CPS) of 10 or more 2.
  • A systematic review and network meta-analysis found that pembrolizumab plus chemotherapy was statistically superior to other immunotherapy- or chemotherapy-based treatment regimens for the first-line treatment of locally recurrent unresectable or metastatic triple-negative breast cancer 3.
  • Pembrolizumab has also been investigated in the neoadjuvant setting for high-risk, early-stage triple-negative breast cancer, with results showing a significant improvement in pathologic complete response rate and 3-year event-free survival compared to neoadjuvant chemotherapy alone 4.

Efficacy and Safety

  • The addition of pembrolizumab to chemotherapy has been shown to result in significantly longer overall survival than chemotherapy alone in patients with advanced triple-negative breast cancer whose tumors express PD-L1 with a CPS of 10 or more 2.
  • The safety profile of pembrolizumab plus chemotherapy has been evaluated in several studies, with common adverse events including neutropenia, febrile neutropenia, and immune-mediated adverse events 2, 5.
  • The impact of pembrolizumab on ovarian function in young triple-negative breast cancer patients treated with chemo-immunotherapy has been evaluated, with results showing no additional impact of pembrolizumab on anti-Müllerian hormone (AMH) evolution compared to chemotherapy alone 6.

Biomarkers and Correlates

  • Tumor PD-L1 expression and stromal tumor-infiltrating lymphocyte (sTIL) levels have been identified as potential biomarkers for response to pembrolizumab in triple-negative breast cancer 2, 5.
  • Higher pre-treatment PD-L1 combined positive score and pre- and on-treatment sTILs have been significantly associated with higher pathologic complete response rates in patients treated with pembrolizumab plus chemotherapy 5.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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