When will I experience side effects from Lutetium-177 (LU-177) infusion?

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Last updated: August 7, 2025View editorial policy

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Side Effects of Lutetium-177 (LU-177) Infusion

Most side effects from Lutetium-177 infusion typically occur within the first few days after treatment, with some immediate reactions possible during infusion and others developing over the following weeks.

Timing of Side Effects

Immediate/During Infusion

  • Infusion reactions may occur during administration or shortly after, though they are relatively uncommon with LU-177 compared to other systemic anticancer therapies 1
  • Symptoms may include flushing, nausea, vomiting, and blood pressure changes 1, 2
  • A physician must remain nearby during administration to monitor for these immediate reactions 1

First 48 Hours

  • Nausea and vomiting are common in the first 1-2 days, primarily due to the amino acid co-infusion rather than the LU-177 itself 2, 3
  • Patients should observe rigorous hygiene during the first 2 days after treatment due to high levels of radioactivity in urine 1, 2

First Week

  • Fatigue commonly occurs within the first week and may persist 2, 4
  • Dry mouth symptoms may begin within the first week 4
  • Radiation protection precautions are most important during the first week 2

2-4 Weeks

  • Hematological side effects typically appear 2-4 weeks after infusion 5, 6
  • Blood count nadirs (lowest points) for neutrophils and platelets typically occur 4-6 weeks post-treatment 5
  • Lymphopenia (decreased lymphocyte count) may be observed around day 15 3

Common Side Effects by System

Gastrointestinal

  • Nausea and vomiting (20-30% of patients) 7, 4
  • Decreased appetite (20-30% of patients) 4
  • Constipation (20% of patients) 4
  • Dry mouth (20-30% of patients) 4

Hematological

  • Anemia (20-30% of patients) 7, 4
  • Thrombocytopenia (2-10% of patients, grade 3-4 in approximately 2%) 7, 5
  • Neutropenia (1-10% of patients, grade 3-4 in approximately 1%) 7, 5
  • Lymphopenia (9-30% of patients) 1, 3

General

  • Fatigue (most common side effect, affecting >20% of patients) 7, 4
  • Electrolyte disturbances (decreased calcium, sodium) 4

Monitoring and Follow-up

  • Complete blood count should be performed every 2-4 weeks after treatment 1
  • Renal and liver function tests should be performed before subsequent cycles 1
  • Long-term follow-up includes blood tests every 8-12 weeks for the first 12 months 1
  • Imaging is typically performed after each cycle to assess treatment response 2

Precautions and Management

  • Adequate hydration is essential before and after treatment (at least 1L of water per day) 2
  • Anti-emetics may be administered prophylactically to manage nausea 2
  • Vital signs should be monitored before and after infusion in symptomatic patients 1
  • Patients should limit close contact with others, particularly children and pregnant women, for several days after treatment 2

Remember that individual responses to LU-177 therapy vary, and your healthcare team will monitor you closely throughout the treatment process. Report any concerning symptoms promptly to your healthcare provider.

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Guideline

Lutetium-177 Infusion Administration

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Research

FDA Approval Summary: Lutetium Lu 177 Vipivotide Tetraxetan for Patients with Metastatic Castration-Resistant Prostate Cancer.

Clinical cancer research : an official journal of the American Association for Cancer Research, 2023

Research

Lutetium-177-PSMA-617 in Low-Volume Hormone-Sensitive Metastatic Prostate Cancer: A Prospective Pilot Study.

Clinical cancer research : an official journal of the American Association for Cancer Research, 2021

Research

Phase 3 Trial of 177Lu-Dotatate for Midgut Neuroendocrine Tumors.

The New England journal of medicine, 2017

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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