What are the instructions for using xylocaine (lidocaine) 5% ointment?

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Instructions for Using Xylocaine 5% Ointment

Apply Xylocaine 5% ointment to the affected area not more than 3 to 4 times daily, and wash hands with soap and water after application. 1

Application Guidelines

Proper Application Technique

  • Apply a thin layer of ointment directly to the affected painful area
  • Use only on intact skin (not on wounds, open sores, or irritated skin)
  • Wash hands thoroughly with soap and water after application
  • For adults and children over 12 years only; consult a doctor for children under 12 1

Timing and Duration

  • Apply no more than 3-4 times daily 1
  • Allow at least 4 hours between applications
  • For optimal anesthetic effect, expect results within approximately 2-5 minutes after application 2
  • Effects typically last 1-2 hours depending on the application site

Specific Uses and Considerations

For Neuropathic Pain

  • Particularly effective for postherpetic neuralgia and other neuropathic pain conditions 3
  • Can be used for dysesthesia (abnormal burning sensations) in vulvodynia or penile dysesthesia 3
  • May be used as first-line treatment before considering systemic medications for localized neuropathic pain 3

For Mucosal Application

  • When used on oral mucosa, a 2-minute application time is typically sufficient to produce adequate analgesia 2
  • For palatal areas, may require up to 5 minutes for optimal effect 2

For Dermatological Procedures

  • Can be applied 20-30 minutes before minor dermatological procedures
  • Provides effective local anesthesia without the need for injections in many cases 4

Safety Precautions

Contraindications

  • Do not use on broken or irritated skin
  • Contraindicated in patients with advanced liver failure due to decreased lidocaine clearance 3
  • Avoid use in patients with known hypersensitivity to amide-type local anesthetics

Potential Side Effects

  • Most common: mild skin reactions such as redness or rash 3
  • Rare but serious: signs of systemic absorption including dizziness, drowsiness, confusion, or seizures
  • If any serious side effects occur, discontinue use and seek medical attention immediately

Special Populations

  • Elderly patients may be more sensitive to effects and side effects
  • Pregnant or breastfeeding women should consult a healthcare provider before use
  • Children under 12 years should use only under medical supervision 1

Important Considerations

Dosage Limitations

  • Do not exceed the recommended frequency of application (3-4 times daily) 1
  • Avoid covering large areas of the body with the ointment to prevent systemic absorption
  • Do not use with occlusive dressings unless specifically directed by a healthcare provider

Storage

  • Store at room temperature away from heat and direct light
  • Keep container tightly closed when not in use
  • Keep out of reach of children

By following these guidelines, Xylocaine 5% ointment can provide effective local pain relief for various conditions while minimizing the risk of adverse effects.

References

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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