What is the investigation of choice for phenylketonuria (PKU) in a newborn?

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Investigation of Choice for Phenylketonuria (PKU) in Newborns

Newborn screening for PKU is performed using tandem mass spectrometry (MS/MS) on dried blood spots collected in the first days of life, followed by confirmatory quantitative plasma amino acid analysis when the screen is positive. 1

Initial Screening Method

Tandem mass spectrometry is now the primary screening method for PKU in the United States, having largely replaced older methods. 1 The three main laboratory methods historically used include:

  • Tandem mass spectrometry (MS/MS) - current standard 1, 2
  • Guthrie bacterial inhibition assay - older method 1
  • Fluorometric analysis - older method 1

MS/MS offers superior accuracy because it simultaneously quantifies both phenylalanine (Phe) and tyrosine (Tyr), allowing calculation of the Phe/Tyr ratio, which dramatically reduces false-positive rates compared to fluorometric methods. 3 Research demonstrates that MS/MS reduces false-positives almost 100-fold when using a Phe/Tyr molar ratio cutoff of 2.5. 3

Confirmatory Diagnostic Testing

When newborn screening is positive, quantitative plasma amino acid analysis is the standard confirmatory method. 1 This analysis must include:

  • Quantitative phenylalanine level 1
  • Phenylalanine-to-tyrosine (Phe:TYR) ratio 1
  • Complete amino acid profile to exclude generalized aminoacidemia 1

Samples should be collected before dietary phenylalanine restriction begins. 1 By the time confirmatory testing occurs, newborns with PAH deficiency typically show phenylalanine concentrations higher than the original screening sample. 1

Critical Additional Testing

Before initiating treatment, tetrahydrobiopterin (BH4) deficiency must be excluded in all newborns with elevated phenylalanine. 1 This is essential because BH4 deficiencies require different treatment approaches. The American College of Medical Genetics recommends:

  • Pterin analysis (neopterin and biopterin) measured in urine or blood 1
  • Erythrocyte dihydropteridine reductase activity measured on whole blood spotted on filter paper 1
  • Quantitative urinary neopterin and biopterin assay to confirm filter paper results 1

Abnormal pterin levels should prompt enzyme testing for deficiencies of GTP cyclohydrolase, 6-pyruvoyl-tetrahydrobiopterin synthetase, dihydropteridine reductase, or pterin carbinolamine-4α-dehydratase. 1

Genotyping for Treatment Planning

PAH genotyping is indicated for improved therapy planning after biochemical diagnosis is confirmed. 1 Genotyping helps determine:

  • The extent of dietary phenylalanine restriction needed 1
  • Likelihood of response to sapropterin (BH4) cofactor supplementation 1
  • Biochemical phenotype severity 4

Timing Considerations

Treatment must begin within the first week of life, with blood phenylalanine in the treatment range by 2 weeks of age to prevent irreversible neurological damage. 1, 2 This requires:

  • Prompt newborn screening (first days of life) 1, 2
  • Rapid follow-up of positive screens 1, 2
  • Immediate confirmatory testing 1
  • Treatment initiation when phenylalanine exceeds 360-605 μmol/L (approximately 6-10 mg/dL) 1

Common Pitfalls to Avoid

Early discharge specimens collected before 24 hours of age have higher false-positive rates with older fluorometric methods, though MS/MS with Phe/Tyr ratio significantly mitigates this issue. 3

Failure to screen for BH4 deficiency before starting dietary treatment is a critical error, as these patients require neurotransmitter replacement therapy rather than dietary restriction alone. 1

Significant variation exists in screening protocols between states, including different cutoff values for positive screens and varying follow-up procedures, which can delay diagnosis. 1, 2

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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