What is the mechanism of action of Depakote (valproate) extended release?

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From the FDA Drug Label

The FDA drug label does not answer the question.

From the Research

Depakote ER (extended-release divalproex sodium) is a long-acting formulation of valproic acid that is effective in treating seizures, bipolar disorder, and migraines, with a dosing range of 500-2000 mg per day, and its use is supported by the most recent study 1.

Key Points

  • Depakote ER is typically taken once daily, with the extended-release formulation maintaining more consistent blood levels throughout the day compared to immediate-release Depakote.
  • The medication works by increasing levels of gamma-aminobutyric acid (GABA) in the brain, which has an inhibitory effect on nerve transmission, helping to stabilize abnormal electrical activity.
  • Common side effects include nausea, drowsiness, dizziness, and weight gain, and regular blood tests are necessary to monitor liver function, platelet counts, and drug levels.
  • Patients should take Depakote ER with food to reduce stomach upset and should not crush or chew the tablets as this would destroy the extended-release mechanism.

Evidence-Based Recommendation

The most recent study 1 found that valproate was more effective than placebo in preventing new bipolar disorder episodes of mania or depression, and not significantly different from lithium, second-generation antipsychotics, or other anticonvulsants.

Clinical Considerations

  • When starting Depakote ER, dosing should be initiated at lower levels and gradually increased to minimize gastrointestinal side effects.
  • The choice of Depakote ER should be based on the patient's history of response and personal preference, as well as the clinician's previous experience and pharmacokinetic properties.
  • Regular monitoring of liver function, platelet counts, and drug levels is necessary to minimize the risk of adverse effects.

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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