What short‑course centrally acting muscle relaxant and dosing is appropriate for a patient with tension‑type headache who has not responded to acetaminophen or NSAIDs?

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Muscle Relaxers for Tension-Type Headache

Direct Answer: Muscle Relaxers Are Not Recommended

There is no evidence supporting the use of centrally acting muscle relaxants for tension-type headache, and current guidelines do not recommend them. 1


Evidence-Based First-Line Treatment

Recommended Acute Medications

  • Ibuprofen 400–800 mg is the most effective first-line treatment for episodic tension-type headache, with superior efficacy compared to acetaminophen or aspirin. 2, 3

  • Acetaminophen 1000 mg provides modest benefit, with a number-needed-to-treat (NNT) of 22 for pain freedom at 2 hours, but is less effective than NSAIDs. 1, 4

  • Naproxen 550–825 mg is an alternative NSAID option with longer duration of action (up to 12 hours). 2

  • Ketoprofen 50–75 mg demonstrates efficacy but may have a higher adverse event rate than other NSAIDs. 2, 3

Combination Therapy for Enhanced Efficacy

  • Adding caffeine to an NSAID or acetaminophen enhances analgesic absorption and provides synergistic pain relief. 5

  • The combination of aspirin 500 mg + acetaminophen 500 mg + caffeine 130 mg is significantly more effective than acetaminophen alone. 6


Critical Frequency Limitation

  • Limit all acute headache medications to ≤2 days per week (≤10 days per month) to prevent medication-overuse headache, which paradoxically increases headache frequency and can lead to daily headaches. 1, 6

When First-Line Treatment Fails

Escalation Algorithm

  1. If acetaminophen fails after 2–3 episodes, switch to an NSAID (ibuprofen 400–800 mg or naproxen 500–825 mg). 6

  2. If NSAIDs fail after 2–3 episodes, consider adding caffeine to the regimen or switching to a different NSAID. 6, 5

  3. If headaches occur >2 days per week, initiate preventive therapy rather than increasing acute medication frequency. 1, 6


Preventive Therapy for Chronic Tension-Type Headache

When to Initiate Prevention

  • Preventive therapy is indicated when headaches occur ≥2 days per week or when acute medication use exceeds the 2-day-per-week threshold. 1, 6

First-Line Preventive Agent

  • Amitriptyline 30–150 mg/day is the only preventive medication with guideline support for chronic tension-type headache, particularly when comorbid depression, anxiety, or sleep disturbances are present. 1, 7

Non-Pharmacologic Options

  • Relaxation therapies with EMG biofeedback and tricyclic antidepressants have similar efficacy rates of 40–50% for chronic tension-type headache. 2

  • Physical therapy and acupuncture are generally less effective than pharmacologic and behavioral interventions. 2


Medications to Avoid

  • Opioids (codeine, hydrocodone, tramadol) are absolutely contraindicated for tension-type headache due to questionable efficacy, high risk of dependence, and precipitation of medication-overuse headache. 7, 6

  • Butalbital-containing compounds should be avoided because they carry a high risk of medication-overuse headache and should be reserved only when all other evidence-based treatments are contraindicated. 7, 8

  • Botulinum toxin injection is not recommended for chronic tension-type headache prevention. 1


Common Pitfalls to Avoid

  • Do not prescribe muscle relaxants (cyclobenzaprine, tizanidine, methocarbamol) for tension-type headache, as they lack evidence of efficacy and are not mentioned in any current guidelines. 1

  • Do not allow patients to use acute medications more frequently in response to treatment failure; instead, transition to preventive therapy. 1, 6

  • Do not substitute one acute medication for another when medication-overuse headache is suspected; instead, withdraw all acute medications and initiate preventive therapy. 7


Red Flags Requiring Urgent Evaluation

  • Seek immediate medical attention if headache includes: thunderclap onset, fever with neck stiffness, progressive worsening pattern, neurological symptoms, or awakening from sleep. 6

References

Guideline

Guideline Directed Topic Overview

Dr.Oracle Medical Advisory Board & Editors, 2025

Research

[Treatment of tension headache].

Revue neurologique, 2000

Research

The use of ibuprofen plus caffeine to treat tension-type headache.

Current pain and headache reports, 2001

Guideline

Alternative Treatment for Headaches When Acetaminophen Fails

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Guideline

Acute Headache Treatment Guidelines

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2026

Guideline

Treatment of Severe Headache with Prednisone

Praxis Medical Insights: Practical Summaries of Clinical Guidelines, 2025

Professional Medical Disclaimer

This information is intended for healthcare professionals. Any medical decision-making should rely on clinical judgment and independently verified information. The content provided herein does not replace professional discretion and should be considered supplementary to established clinical guidelines. Healthcare providers should verify all information against primary literature and current practice standards before application in patient care. Dr.Oracle assumes no liability for clinical decisions based on this content.

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