How are glucopeptides classified pharmacologically?

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From the Research

Los glucopeptidos se clasifican farmacológicamente como secretagogos de insulina que estimulan la liberación de insulina en el páncreas. Estos medicamentos, como la repaglinida y la nateglinida, pertenecen a la clase de meglitinidas y actúan inhibiendo los canales de potasio sensibles a ATP en la membrana de las células beta del páncreas, lo que lleva a una liberación rápida de insulina [ 1 ].

Algunos de los beneficios de los glucopeptidos incluyen:

  • Una acción rápida y breve, lo que reduce el riesgo de hipoglucemia [ 2 ]
  • Eficacia en el control de la glucemia posprandial [ 3 ]
  • Pueden ser utilizados en combinación con otros medicamentos orales para el tratamiento de la diabetes tipo 2 [ 4 ]
  • Son una opción para pacientes con diabetes tipo 2 que requieren una mayor flexibilidad en su tratamiento [ 5 ]

Es importante destacar que, aunque los glucopeptidos son efectivos en el control de la glucemia, su uso debe ser evaluado cuidadosamente en cada paciente, considerando factores como la edad, la función renal y la presencia de otras enfermedades [ 1 ].

References

Research

Insulin secretagogues: who, what, when, and how?

Current diabetes reports, 2005

Research

Oral hypoglycemic agents: insulin secretagogues, alpha-glucosidase inhibitors and insulin sensitizers.

Experimental and clinical endocrinology & diabetes : official journal, German Society of Endocrinology [and] German Diabetes Association, 2001

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